Didesmethyl cariprazine

二去甲基卡利拉嗪

SCHEMBL3409190 | SCHEMBL1302192 | UNII-6AY300X9G3 | Didesmethyl cariprazine | DDCAR | [4-[2-[4-(2,3-dichlorophenyl)piperazin-1-yl]ethyl]cyclohexyl]urea | Urea, N-(trans-4-(2-(4-(2,3-dichlorophenyl)-1-piperazinyl)ethyl)cyclohexyl)- | AKOS040741633 | HY-100

Didesmethyl cariprazine

D651098-5mg

5mg

≥99%

-20°C储存

超低温冰袋运输

Didesmethyl cariprazine is a metabolite of Cariprazine and acts as the predominant circulating active moiety. Didesmethyl cariprazine has a long half-life of 1-3 weeks. Cariprazine is a antipsychotic agent candidate that exhibits high affinity for the D 3 and D 2 receptors, and moderate affinity for the 5-HT 1A receptor Form:Solid IC50& Target:5-HT 1A Receptor D 3 Receptor D 2 Receptor

双甲基卡哌嗪是卡哌嗪的代谢物，是主要的循环活性分子。双甲基卡哌嗪的半衰期较长，为 1-3 周。卡利普嗪是一种抗精神病候选药物，对 D 3

839712-25-3

C19H28Cl2N4O

399.36 g/mol

11200383

C1CC(CCC1CCN2CCN(CC2)C3=C(C(=CC=C3)Cl)Cl)NC(=O)N

[4-[2-[4-(2,3-dichlorophenyl)piperazin-1-yl]ethyl]cyclohexyl]urea

1S/C19H28Cl2N4O/c20-16-2-1-3-17(18(16)21)25-12-10-24(11-13-25)9-8-14-4-6-15(7-5-14)23-19(22)26/h1-3,14-15H,4-13H2,(H3,22,23,26)

UMTWXZNVNBBFLC-UHFFFAOYSA-N

C1CC(CCC1CCN2CCN(CC2)C3=C(C(=CC=C3)Cl)Cl)NC(=O)N

11200383

839712-25-3

DMSO : 11.36 mg/mL (28.45 mM; ultrasonic and warming and heat to 80°C)

2

3

5

398.164 Da

398.164 Da

61.600 Ų

26

0

451

0

1

3.7