Galantide TFA

加兰肽TFA

Galantide TFA

G659296-5mg

5mg

≥98%

避光,充氩,干燥,-80℃储存

超低温冰袋运输

Galantide TFA is a reversible and non-specific galanin (GAL) receptor antagonist. Galantide TFA dose-dependently shows antagonism to galanin-induced K + conductance with an IC 50 value of 4 nM. Galantide TFA can be used for the research of neurological di Appearance:Solid In Vitro:Galantide TFA (0.1-10000 nM) inhibits the galanin-induced activation of the K + conductance with an IC 50 value of 4 nM. Galantide TFA (0.1-10000 nM) dose-dependently inhibits the voltage-dependent Ba 2+ current with an IC 50 value of 16 nM. Gal In Vivo:Galantide TFA (5 nm; icv, once) inhibits luteinizing hormone (LH) release of ovariectomized (OVX) rats. Galantide TFA (1 and 5 nm; iv, for 3 times, at 1300, 1400 and 1500 h) decreases steroid-induced luteinizing hormone (LH) surge in estradiol benzoa Biological Activity:Galantide TFA is a reversible and non-specific galanin (GAL) receptor antagonist. Galantide TFA dose-dependently shows antagonism to galanin-induced K + conductance with an IC 50 value of 4 nM. Galantide TFA can be used for the research of neurological di

C106H152F3N25O28S

2313.55 g/mol

DMSO : 100 mg/mL (43.22 mM; Need ultrasonic) H2O : < 0.1 mg/mL (ultrasonic;adjust pH to 2 with HCl) (insoluble)