LAS101057, 腺苷 A2b 受体拮抗剂

LAS101057

L656526-1ml

1ml

10mM in DMSO

避光,-80℃储存

超低温冰袋运输

LAS101057 is a potent, selective, and orally efficacious A2B receptor antagonist. In Vivo At 3 mg/kg, LAS101057 is active in preventing Acetyl-β-methylcholine-induced AHR, and at 10 mg/kg it inhibits AHR to Acetyl-β-methylcholine to a level virtually equal to that seen with Hexadecadrol at 1 mg/kg . MCE has not independently confirmed the accuracy of these methods. They are for reference only.

LAS101057 是一种强效、选择性和口服有效的 A2B 受体拮抗剂。

925676-48-8(DMSO)

C18H14FN5O

335.34 g/mol

FC1=CN=CC=C1C(N=CC(NC(C2CC2)=O)=N3)=C3C4=CC=CN=C4

拮抗剂

腺苷 A2b 受体拮抗剂