(+)-Penbutolol

(+)-喷布洛尔

CCRIS 2854 | HY-116790A | KQXKVJAGOJTNJS-OAHLLOKOSA-N | MS-24164 | (+)-Isopenbutolol | 2-Propanol, 1-(2-cyclopentylphenoxy)-3-((1,1-dimethylethyl)amino)-, (R)- | (2r)-1-(tert-butylamino)-3-(2-cyclopentylphenoxy)propan-2-ol | AKOS040740652 | SCHEMBL1652319

(+)-Penbutolol

P651513-5mg

5mg

≥95%

-20°C储存

超低温冰袋运输

(+)-Penbutolol is a β-adrenoceptor antagonist, with an IC 50 of 0.74 μM (+)-Penbutolol is an optical isomer of l-penbutolol with Na + channel-blocking action . In Vitro (+)-penbutolol on the [Ca 2+ ] i -increase induced by LPC is concentration-dependent. (+)-penbutolol inhibits the rounding of cells dose dependently (8±4%, 56±4% and 66±2% at the concentrations of 10 -6 M, 5×10 -6 M and 10 -5 M, respectively). MCE has not independently confirmed the accuracy of these methods. They are for reference only. Form:Solid IC50& Target:IC50: 0.74 μM (β-adrenoceptor)

(+)-Penbutolol 是一种 β 肾上腺素受体拮抗剂，IC50 为 0.74 μM。(+)-Penbutolol 是 l-penbutolol 的光学异构体，具有阻断 Na + 通道的作用。

38363-41-6

C18H29NO2

291.43 g/mol

162302

CC(C)(C)NC[C@H](COC1=CC=CC=C1C2CCCC2)O

(2R)-1-(tert-butylamino)-3-(2-cyclopentylphenoxy)propan-2-ol

1S/C18H29NO2/c1-18(2,3)19-12-15(20)13-21-17-11-7-6-10-16(17)14-8-4-5-9-14/h6-7,10-11,14-15,19-20H,4-5,8-9,12-13H2,1-3H3/t15-/m1/s1

KQXKVJAGOJTNJS-OAHLLOKOSA-N

CC(C)(C)NCC(COC1=CC=CC=C1C2CCCC2)O

162302

38363-41-6

DMSO : 100 mg/mL (343.14 mM; Need ultrasonic)

2

3

7

291.22 Da

291.22 Da

41.500 Ų

21

0

294

0

1

4.2