RIPK1-IN-4

小分子

RIPK1-IN-4

R655286-1ml

1ml

10mM in DMSO

-80℃储存

超低温冰袋运输

RIPK1-IN-4 (compound 8) is a potent and selective type II kinase inhibitor of receptor interacting protein 1 (RIP1) kinase and binds to a DLG-out inactive form of RIP1 with an IC 50 s of 16 nM and 10 nM for RIP1 and ADP-Glo kinase IC50& Target:IC50: 16 nM (RIP1) and 10 nM (ADP-Glo)

RIPK1-IN-4 （化合物 8）是受体互作蛋白 1（RIP1）激酶的一种强效、选择性 II 型激酶抑制剂，能与 DLG-out 非活性形式的 RIP1 结合，对 RIP1 和 ADP-Glo 激酶的 IC 50 s 分别为 16 nM 和 10 nM。

1481641-08-0(DMSO)

C23H23N5O2

401.46 g/mol

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