NCT-501是一种有效的选择性Aldehyde Dehydrogenase 1A1 (ALDH1A1)抑制剂，IC50为40 nM。 Information NCT-501 NCT-501 is a potent and selective inhibitor of Aldehyde Dehydrogenase 1A1 (ALDH1A1) with IC50 of 40 nM. Targets ALDH1A1 40 nM In vitro In Caco-2 cell line, NCT-501 exhibits excellent permeability. In vivo In CD1 Mice, NCT-501 is well absorbed and distributed but rapidly metabolized and/or excreted.