Ilmofosine 是具有抗肿瘤活性的PKC抑制剂，IC 50为560 nM。它在PKC的调控位点起竞争性抑制剂的作用。浓度为1-30μg/ mL的伊莫福辛具有抗多种人类非小细胞肺癌，乳腺癌，结肠直肠癌，卵巢癌和肾细胞癌的功效。 Ilmofosine is a PKC inhibitor with antineoplastic activity with an IC|50|value of 560 nM. It acts as a competitive inhibitor at the regulatory site of PKC. Ilmofosine has efficacy against various human non-small cell lung, breast, colorectal, ovarian, and renal cell cancers at concentrations of 1-30 μg/mL.